I. Paper
| 1 | Design and Synthesis of Ether Derivatives of Spliceostatin A and their Biological Evaluation towards Prostate Cancer Treatment Satoru Hirabayashi, Yue Li, Noriko Ohta, Airi Ishibashi, YusukeYoshikawa, Bangzhong Lin, Megumi Fumimoto, Tsunayoshi Takehara, Kazuto Nunomura, Takeyuki Suzuki, Junichi Haruta, Keisuke Nimura, Mitsuhiro Arisawa* Tetrahedron Lett. 2023, 114, 154288. DOI: 10.1016/j.tetlet.2022.154288   |
| 2 | A New Tetracyclic Bromopyrrole-Imidazole Derivative through Direct Chemical Diversification of Substances Present in Natural Product Extract from Marine Sponge Petrosia (Strongylophora) sp. Natchanun Sirimangkalakitti, Kazuo Harada, Makito Yamada, Masayoshi Arai*, Mitsuhiro Arisawa* Molecules 2023, 28, 143. (INVITED) DOI: 10.3390/molecules28010143  |
| 3 | Reagent-Controlled Regioselective Intramolecular [2+2] Cycloaddition between Vinylsilanes and Allenes Shohei Yoshioka, Tsunayoshi Takehara, Takeyuki Suzuki, Mitsuhiro Arisawa* Chem. Eur. J. 2023, 29, e202203556. DOI: 10.1002/chem.202203556  |
| 4 | Electrochemical Synthesis of Hetero[7]helicenes Containing Pyrrole and Furan Rings via an Oxidative Heterocoupling and Dehydrative Cyclization Sequence Mohamed S. H. Salem, Md. Imrul Khalid, Makoto SAKO, Keigo Higashida, Charlie Lacroix, Masaru Kondo, Ryo Takishima, Taisei Taniguchi, Masahiro Miura, Giang Vo-Thanh, Hiroaki Sasai, Shinobu Takizawa* Adv. Synth. Catal. 2023, 365, 373–380. DOI: 10.1002/adsc.202201262  |
| 5 | Absorption, fluorescence, and two-photon excitation ability of 5-phenyl-13-arylisoindolo[2,1-a]quinolines prepared by one-pot reaction of ring-closing metathesis and 1,3-dipolar cycloaddition Avena Francisco Ramon, Yuki Wada, Hirokazu Ishii, Yuki Watakabe, Motosuke Tsutsumi, Kwangkyun Jang, Kohei Otomo, Lin Qiao, Yuki Fujii, Hirofumi Tsujino, Yasuo Tsutsumi, Tomomi Nemoto, Mitsuhiro Arisawa* Dyes and Pigments 2023, 212, 111118. DOI: 10.1016/j.dyepig.2023.111118 2025年3月24日まで無料ダウンロード可能 https://www.sciencedirect.com/science/article/pii/S0143720823000438?dgcid=author
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| 6 |
Palladium-Catalyzed Intramolecular Migratory Cycloisomerization of 3-Phenoxy Acrylic Acid Ester via C–O Bond Cleavage and C–O/C–C Bonds Formation for 2,3-Disubstituted Benzofurans Synthesis
Yuichi Kuboki, Shohei Ohno, Makoto Sako, Kenichi Murai, Mitsuhiro Arisawa*
Chem. Pharm. Bull. 2023, 71, 93–100. (INVITED)
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| 7 |
Ligand-free Reductive Coupling of Aldehyde with 1,3-diene Using Sulfur-Modified Au-Supported Nickel Nanoparticle Catalyst
Ryosuke Ohta#, Yasunori Shio#, Toshiki Akiyama, Makito Yamada, Kazuo Harada and Mitsuhiro Arisawa*
# equal contribution
New J. Chem. 2023, 47, 7694-7700.
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| 8 | Design and Synthesis of 4-Acetoxypentanamide Derivatives of Spliceostatin A and Their Biological Evaluation towards Prostate Cancer Treatment Satoru Hirabayashi, Yuko Tsuyuguchi, Yue Li, Noriko Ohta, Yusuke Yoshikawa, Bangzhong Lin, Megumi Fumimoto, Kazuto Nunomura, Takeyuki Suzuki, Junichi Haruta, Keisuke Nimura, Mitsuhiro Arisawa* Bioorg. Med. Chem. Lett. 2023, 91, 129333. DOI: 10.1016/j.bmcl.2023.129333
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| 9 | Synthesis and Biological Evaluation of Simplified Ansellone Analogues with Lipophilic Side Chains as HIV-Latency-Reversing Agents Mizushi Yanagihara, Naoki Kishimoto, Kanae Nakahara, Towa Abe, Satoshi Miura, Bangzhong Lin, Megumi Fumimoto, Junichi Haruta, Shogo Misumi, Mitsuhiro Arisawa*, Kenichi Murai* Chem. Eur. J. 2023, e202300677. DOI:10.1002/chem.202300677
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| 10 | Heteroannulation of Bicyclobutane Derivatives via Au-catalyzed Hydration to Enol Ethers and Intramolecular Cyclization Giving Spirocyclobutanes Masaharu Takatsuki, Hiroshi Aoyama, Kenichi Murai, Mitsuhiro Arisawa*, Makoto Sako* Chem. Commun. 2023, 59, 7467-7470. DOI: 10.1039/D3CC01955A  |
| 11 | Development of Cycloisomerization with Rearrangement of a Tosyl Group Using N-Tosyl-o-allenylaniline Shohei Yoshioka, Masaharu Takatsuki, Tsunayoshi Takehara, Takeyuki Suzuki, Mitsuhiro Arisawa* J. Org. Chem. 2023, 88, 11268–11277. DOI: 10.1021/acs.joc.3c00625  |
| 12 | A versatile Plasmodium falciparum reporter line expressing NanoLuc enables highly sensitive multi-stage drug assays Yukiko Miyazaki*, Martijn W. Vos, Fiona J. A. Geurten, Pierre Bigeard, Hans Kroeze, Shohei Yoshioka, Mitsuhiro Arisawa, Daniel Ken Inaoka, Valerie Soulard, Koen J. Dechering, Blandine Franke-Fayard, Shinya Miyazaki* Nature Portfolio Communications Biology 2023, 6, 713 DOI: 10.1038/s42003-023-05078-5長崎大学と大阪大学が共同プレスリリースしました。 https://www.nagasakiu.ac.jp/ja/guidance/kouhou/press/file/2023/20230721-1-1.pdf https://resou.osaka-u.ac.jp/ja/research/2023/20230721_1
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| 13 | Axially Chiral Borinic Acid Catalysts: Design, Synthesis, and Application in Alkylative Desymmetrization of 1,2-Diols Yuta Chikashige, Tsunayoshi Takehara, Tsuyoshi Matsuzaki, Takeyuki Suzuki, Kenichi Murai, Mitsuhiro Arisawa*, Makoto Sako* J. Org. Chem. 2023, 88, 14178-14183. DOI: 10.1021/acs.joc.3c01143  |
| 14 | Data-driven Electrochemical One-pot Synthesis of Double Hetero[7]dehydrohelicene Mohamed S. H. Salem*, Rubal Sharma, Md. Imrul Khalid, Meghna Sasi, Ryo Amasaki, Yoshitane Imai, Mitsuhiro Arisawa, Shinobu Takizawa* Electrochemistry, 2023, in press. DOI: 10.5796/electrochemistry.23-67092  |
II. Review
| 1 | ファーマシスト・サイエンティストの養成 有澤光弘 薬学教育 2023, in press DOI：10.24489/jjphe.2023-018  |
III. Winning Prize
| 1 | 日本薬学会第143年会 学生優秀発表賞 吉岡くん（D4）が日本薬学会 第143年会で優秀発表賞（口頭発表）を受賞しました。 |
| 2 | 第26回ヨウ素学会シンポジウム 優秀ポスター賞 髙島さん（B5）が第26回ヨウ素学会シンポジウムで優秀ポスター賞を受賞しました。 |
IV. その他
| 1 | 2023.03.13 髙月君（M2）が公益財団法人 吉田科学技術財団 国際研究集会派遣研究者事業に採択されました。 |