大阪大学薬学部 医薬合成化学分野

2008 Publications

1 Oxidative Cross-Coupling of Arenes Leading to Biaryls by Use of Organo-
Iodine(III) Oxidants
T. Dohi, M. Ito, K. Morimoto, M. Iwata
Angew. Chem. Int. Ed., 47, 1301-1304 (2008)
2 A Chiral Hypervalent Iodine (III) Reagent for Enantioselective Dearomatization of Phenols
T. Doi, A. Maruyama, N. Takenaga, K. Senami, Y. Minamitsuji, H. Fujioka, Simon B. Caemmerer, Y. Kita
Angew. Chem. Int. Ed., 47, 3787-3790 (2008)
3 Facile Formation of Tetrahedrofurans with Multiple Chiral Centers using Double Iodoetherification ofσ- Symmetric Diene Acetals: Short Asymmetric Total Synthesis of Rubrenolide and Rubrynolide
H. Fujioka, Y. Ohba, H. Hirose, K. Nakahara, K. Murai, Y. Kita
Tetrahedron, 64, 4233-4245 (2008)
4 A New H2O2/Acid anhydride system for the
iodoarene-catalyzed C-C bond-forming reactions of Phenols T. Dohi, Y. Minamitsuji, A. Maruyama, S. Hirose, Y. Kita ;
.Organic Lett.,10,3559-3562 (2008)
5 Clean and Efficient Benzylic C-H Oxidation in Water Using a Hypervalent Iodine Reagent: Activation of Polymeric Iodosobenzene with KBr in the Presence of Montmorillonite-K10
Dohi T, Takenaga N, Goto A, Fujioka H, Kita Y
J. Org. Chem., 73, 7365-7368 (2008)
6 Oxidative decarboxylative synthesis of 2-H-imidazolines from glyoxylic acid and 1,2-diamines;
Murai K, Morishita M, Nakatani R, Fujioka H, Kita Y
Chem Commun., 4498-4500 (2008)
Synthesis of biaryl compounds through three-component assembly: ambidentate effect of the tert-butyldimethylsilyl group for regioselective Diels-Alder and Hiyama coupling reactions
Akai S, Ikawa T, Takayanagi S, Morikawa Y, Mohri S, Tsubakiyama M, Egi M, Wada Y, Kita Y
Angew. Chem. Int. Ed., 47, 7673-7676 (2008)
8 One-pot three-component reaction providing 1,5-benzodiazepine derivatives
Murai K, Nakatani R, Kita Y, Fujioka H
Tetrahedron, 64, 11034-11040 (2008)

総説

1 超原子価ヨウ素の化学の新展開とグリーンケミストリー
北 泰行
化学工業, 59, 16-22 (2008)
2 アセタール脱保護の新手法-ケタールの存在下にアセタールを加水分解する-
藤岡弘道、北 泰行
医薬品原薬・中間体製造におけるスケールアップとトラブル対策 (CMC出版), 194-209 (2008)

著書

1 Syntheses of anthracyclines and fredericamycin A via strong base-induced cycloaddition reaction of homophthalic anhydrides
Kita Y, Fujioka H Top. Curr. Chem.,
282 (Anthracycline Chemistry and Biology I), 299-319 (2008)