| I. | Paper |
| 1 | An Entry to Chiral 1,1,2,3-Tetrasubstituted Arylcyclopropanes by Pd(II)-Catalyzed Arylation via Directing Group-Mediated C(sp3)-H Activation Naoyuki Hoshiya, Moemi Kondo, Hayato Fukuda, Mitsuhiro Arisawa, Jun’ichi Uenishi, and Satoshi Shuto. J. Org. Chem. 2017,82, 535–2544. DOI:10.1021/acs.joc.6b02935  |
| 2 | Cyclopropane-Based Peptidomimetics Mimicking Wide-Ranging Secondary Structures of Peptides: Conformational Analysis and Their Use in Rational Ligand Optimization Akira Mizuno, Tomoshi Kameda, Tomoki Kuwahara, Hideyuki Endoh, Yoshihiko Ito, Shizuo Yamada, Kimiko Hasegawa, Akihito Yamano, Mizuki Watanabe, Mitsuhiro Arisawa, Satoshi Shuto. Chem. Eur. J. 2017, 23, 3156-3168. DOI: 10.1002/chem.201605312  |
| 3 | First Asymmetric Total Synthesis and Insight into the Structure of Laurenidificin Yusuke Yoshikawa, Maki Yamakawa, Tetsuya Kobayashi, Kunio Suzuki, Mitsuhiro Arisawa, Hiromichi Fujioka. Eur. J. Org. Chem. 2017, 19, 2715-2718.DOI: 10.1002/ejoc.201700321  |
| 4 | Cycloisomerization between Aryl Enol Ether and Silylalkynes under Ruthenium Hydride Catalysis: Synthesis of 2,3-Disubstituted Benzofurans Shohei Ohno, Kohei Takamoto, Hiromichi Fujioka, Mitsuhiro Arisawa Org. Lett. 2017, 19, 2422-2425.DOI: 10.1021/acs.orglett.7b00985  |
| 5 | One-pot Enyne Metathesis/Diels–Alder/Oxidation to Six-membered Silacycles with a Multi-ring Core: Discovery of Novel Fluorophores Shohei Yoshioka, Yuki Fujii, Hirofumi Fujino, Tadayuki Uno, Hiromichi Fujioka, Mitsuhiro Arisawa Chem. Commun. 2017, 53, 5970-5973. DOI: 10.1039/C7CC02788E  |
| 6 | Ligand-Free Suzuki–Miyaura Coupling Using Ruthenium(0) Nanoparticles and a Continuously Irradiating Microwave System Toshiki Akiyama, Takahisa Taniguchi, Nozomi Saito, Ryohei Doi, Tetsuo Honma, Yusuke Tamenori, Yuuta Ohki, Naoyuki Takahashi, Hiromichi Fujioka, Yoshihiro Sato, Mitsuhiro Arisawa Green Chem. 2017, 19, 3357-3369.DOI: 10.1039/C7GC01166K  |
| 7 | Concise synthesis of oxacyclic compounds using highly discriminative two-way transformations of α,β-unsaturated esters in the presence of enones Kenta Morita, Reiya Ohta, Hiroshi Aoyama, Kenzo Yahata, Mitsuhiro Arisawa, Hiromichi Fujioka Chem. Commun. 2017, 53, 6605-5508. DOI: 10.1039/C7CC03287K  |
| 8 | Transformation of Methylene Acetals to Bromoformates with a Combination of Trimethyl(phenylthio)silane and N-Bromosuccinimide Satoshi Takano, Takayoshi Tsuzuki, Takashi Murayama, Tomoshi Kameda, Yasuhiro Kumaki, Takashi Sakurai, Hayato Fukuda, Mizuki Watanabe, Mitsuhiro Arisawa, Satoshi Shuto J. Med. Chem. 2017, 60, 5868-5875.DOI: 10.1021/acs.jmedchem.7b00540 |
| 9 | Synthesis of 8-Substituted Analogues of Cyclic ADP-4-Thioribose and Their Unexpected Identification as Ca2+-Mobilizing Full Agonists Tomohiro Megawa, Misa Nogata, Yuuka Hirose, Shun Ohgami, Akira Nakamura, Yasuyoshi Miki, and Hiromichi Fujioka J. Org. Chem., 2017, 82 (14), pp 7608–7613.DOI: 10.1021/acs.joc.7b00776 |
| 10 | Ruthenium-Catalyzed 1,6-Aromatic Enamide−Silylalkyne Cycloisomerization: Approach to 2,3-Disubstituted Indoles Kohei Takamoto, Shohei Ohno, Norimichi Hyogo, Hiromichi Fujioka, and Mitsuhiro Arisawa J. Org. Chem. 2017, 82. 8733-8742. DOI: 10.1021/acs.joc.7b01288  |
| 11 | Versatile and chemoselective synthesis of fluorinated methyl ethers from methoxymethyl ethers Reiya Ohta, Yuichi Kuboki, Yuki Yoshikawa, Yasuyuki Koutani, Tomohiro Maegawa, Hiromichi Fujioka Journal of Fluorine Chemistry, 2017, 201, 1-6.DOI:org/10.1016/j.jfluchem.2017.07.007  |
| 12 | Synthesis of 8-Substituted Analogues of Cyclic ADP-4-Thioribose and Their Unexpected Identification as Ca2+-Mobilizing Full Agonists Satoshi Takano, Takayoshi Tsuzuki, Takashi Murayama, Tomoshi Kameda, Yasuhiro Kumaki, Takashi Sakurai, Hayato Fukuda, Mizuki Watanabe, Mitsuhiro Arisawa, Satoshi Shuto Journal of Medicical Chemistry, 2017, 60, 5868-5875.DOI:10.1021/acs.jmedchem.7b00540  |
| 13 | Transformation of Methylene Acetals to Bromoformates with a Combination of Trimethyl(phenylthio)silane and N-Bromosuccinimide Tomohiro Maegawa, Misa Nogata, Yuuka Hirose, Shun Ohgami, Akira Nakamura, Yasuyoshi Miki, Hiromichi Fujioka Journal of Organic Chemistry, 2017, 82, 7608-7613.DOI:10.1021/acs.joc.7b00776  |
| 14 | Enantio- and Diastereoselective Betti/aza-Michael Sequence: Single Operated Preparation of Chiral 1,3-Disubstituted Isoindolines Shinobu Takizawa, Makoto Sako, Mohamed Ahmed Abozeid, Kenta Kishi, H. D. P. Wathsala, Shuichi Hirata, Kenichi Murai, Hiromichi Fujioka, Hiroaki Sasai Organic Letters, 2017, 19, 5426–5429.DOI:10.1021/acs.orglett.7b02693  |
| II. | Review |
| 1 | エナミドメタセシス反応を用いたインドメタシン誘導体の合成と多剤耐性抗がん剤への展開 Mitsuhiro Arisawa Biophila 2017, 6, 29-39. |
| 2 | Chemoselective reduction and alkylation of carbonyl functions using phosphonium salts as an in situ protecting groups Reiya Ohta, Hiromichi Fujioka Chem. Pharm. Bull. 2017, 65, 10-18.  |
| Ⅲ. | Winning Prize |
| 1 | 第43回反応と合成の進歩シンポジウム・富山学生ポスター賞受賞 M2の窪木さんが富山学生ポスター賞を受賞されました。おめでとうございます。 http://www.43spors.jp/common/pdf/winning/student_poster.pdf |
| 2 | 大阪大学賞受賞 有澤准教授が平成29年度大阪大学賞を受賞することになりました。 http://www.phs.osaka-u.ac.jp/information/topics_detail.cgi?id=1511758954 |