大阪大学薬学部 医薬合成化学分野

2018 Publications

 

 

I. Paper
1 Aromatic aldehyde-selective aldol addition with aldehyde-derived silyl enol ethers
Takahiro Kawajiri, Reiya Ohta, Hiromichi Fujioka, Hironao Sajiki, Yoshinari Sawama
Chem. Commun. 2018, 54, 374-377.
DOI:10.1039/C7CC08936H
Graphical abstract: Aromatic aldehyde-selective aldol addition with aldehyde-derived silyl enol ethers
2 Palladium-Catalyzed Seven-Membered Silacycle Construction: 1,7-Enyne Hydroxycyclization To Give a Benzosilepine Skeleton
Kohei Takamoto, Shohei Yoshioka, Hiromichi Fujioka, Mitsuhiro Arisawa
Org. Lett. 2018, 20, 1773-1776.
DOI:10.1021/acs.orglett.8b00271
3 Selective Transformation of β‐Disubstituted Enones and Ynones in the Presence of β‐Monosubstituted Enones
Kenta Morita, Reiya Ohta, Kei Watanabe, Hiromichi Fujioka
Asian J. Org. Chem. 2018, 7, 829–835.
DOI:org/10.1002/ajoc.201700711
4 Oxidative Rearrangement of Secondary Amines Using Hypervalent Iodine(III) Reagent
Kenichi Murai, Tetsuya Kobayashi, Makoto Miyoshi, Hiromichi Fujioka
Org. Lett. 2018, 20, 2333-2337.
DOI:10.1021/acs.orglett.8b00675
5 Highly Discriminative and Chemoselective Deprotection/Transformations of Acetals with the Combination of Trialkylsilyl Triflate/2,4,6-Collidine
Reiya Ohta, Nao Matsumoto, Yoshifumi Ueyama, Yuichi Kuboki, Hiroshi Aoyama, Kenichi Murai, Mitsuhiro Arisawa, Tomohiro Maegawa, Hiromichi Fujioka
J. Org. Chem. 2018, 83, 6432–6443.
DOI:10.1021/acs.joc.8b00675
6 Cascade Multiple Diels–Alder Reactions of Styrene Derivatives with Maleimide or Maleic Anhydride
Shohei Yoshioka, Hiroshi Aoyama, Hiromichi Fujioka, Mitsuhiro Arisawa
J. Org. Chem. 2018, 83, 6599–6606.
DOI:10.1021/acs.joc.8b00890
7 Synthesis of Chiral cis-Cyclopropane Bearing Indole and Chromone as Potential TNFα Inhibitors
Ryutaro Kanada, Makoto Tanabe, Ryuta Muromoto, Yukina Sato, Tomoki Kuwahara, Hayato Fukuda, Mitsuhiro Arisawa, Tadashi Matsuda, Mizuki Watanabe, Satoshi Shuto
J. Org. Chem. 2018, 83, 7672–7682.
DOI:10.1021/acs.joc.8b00466
8 Design and synthesis of histamine H3/H4 receptor ligands with a cyclopropane scaffold
Mizuki Watanabe, Takaaki Kobayashi, Yoshihiko Ito,Hayato Fukuda, Shizuo Yamada, Mitsuhiro Arisawa, Satoshi Shuto
Bioorg. Med. Chem. Lett. 2018, 28, 3630-3633.
DOI:org/10.1016/j.bmcl.2018.10.041
9 Reusable Immobilized Iron(II) Nanoparticle Pre-Catalysts for Ligand-Free Kumada Coupling
Toshiki Akiyama, Yuki Wada, Kellie Jenkinson, Tetsuo Honma, Kazuki Tsuruta, Yusuke Tamenori, Hitoshi Haneoka, Tsunayoshi Takehara, Takeyuki Suzuki, Kenichi Murai, Hiromichi Fujioka, Yoshihiro Sato, Andrew E. H. Wheatley, Mitsuhiro Arisawa
ACS Appl. Nano Mater. 2018, 1, 6950–6958.
DOI:10.1021/acsanm.8b01742
II. Review
Ⅲ. Winning Prize
1 2018 Filipino Scholars Symposium at Osaka University ポスター賞(金賞)
M1のAvena Ramonさんが2018 Filipino Scholars Symposium at Osaka Universityにてポスター賞(金賞)を受賞されました。おめでとうございます。
http://www.phs.osaka-u.ac.jp/information/topics_detail.cgi?id=1545891380
Ⅳ. Book
1 天然有機分子の構築:全合成の魅力(化学の要点シリーズ)
日本化学会 編・中川昌子・有澤光弘 著
共立出版
ISBN 978-4-320-04467-8