大阪大学薬学部 医薬合成化学分野

2022 Publications

 

I.

Paper

1

Doubleisomerization / cycloisomerization / aromatization of 1-(allyloxy)-2-(cyclopropylmethyl)benzenes to give 2-ethyl-3-isopropylbenzofurans using multitasking single rhodium catalyst
Yuta Sato, Tsuyoshi Matsuzaki, Tsunayoshi Takehara, Makoto Sako, Mitsuhiro Arisawa*
Chem. Commun.  2022, 58, 415-418.
DOI: 10.1039/D1CC06163A
Graphical abstract: Double isomerization/cycloisomerization/aromatization of 1-(allyloxy)-2-(cyclopropylmethyl)benzenes to give 2-ethyl-3-isopropylbenzofurans using a multitasking single rhodium catalyst
2 Metal-free C(aryl)–P Bond Cleavage: Experimental and Computational Studies of the Michael Addition/aryl migration of Triarylphosphines to Alkynyl Esters
Makoto Sako, Kyohei Kanomata, Mohamed S. H. Salem, Tomohiro Furukawa, Hiroaki Sasai, Shinobu Takizawa*
Org. Chem. Front. 2022, 9, 2187-2192.
DOI: 10.1039/D2QO00028H
3 Carbon(sp2)-carbon(sp3) Bond-forming Cross-coupling Reactions Using Sulfur-Modified Au-Supported Nickel Nanoparticle Catalyst
Ryosuke Ohta, Yasunori Shio, Toshiki Akiyama, Makito Yamada, Shuhei Shimoda, Kazuo Harada, Makoto Sako, Jun-ya Hasegawa, Mitsuhiro Arisawa*
Asian J. Org. Chem. 2022, 11, e202200229.
DOI: 10.1002/ajoc.202200229
Description unavailable
4 Design, Synthesis, and Monoamine Oxidase B Selective Inhibitory Activity of N-Arylated Heliamine Analogues
Makito Yamada, Yu Hirose, Bangzhong Lin, Megumi Fumimoto, Kazuto Nunomura, Sirimangkalakitti Natchanun, Naoyuki Takahashi, Yuuta Ohki, Makoto Sako, Kenichi Murai, Kao Harada, Masayoshi Arai, Sayo Suzuki, Tomonori Nakamura, Junichi Haruta, Mitsuhiro Arisawa*
ACS Med. Chem. Lett. 202213, 1582–1590.
DOI: 10.1021/acsmedchemlett.2c00228
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5

Substrate-Assisted Reductive Elimination Determining the Catalytic Cycle: A Theoretical Study on the Ni-Catalyzed 2,3-Disubstituted Benzofuran Synthesis via CO Bond Activation
Ray Miyazaki, Kenji Iida, Shohei Ohno, Tsuyoshi Matsuzaki, Takeyuki Suzuki, Mitsuhiro Arisawa, Jun-ya Hasegawa*
Organometallics ASAP
DOI: 10.1021/acs.organomet.2c00419

6 Double rearrangement strategy for fused 3-benzazepines: Alternative synthesis of the Dolby–Weinreb enamine
Saito Keigo, Aoyama Hiroshi, Sako Makoto, Arisawa Mitsuhiro*, Murai Kenichi*
J. Org. Chem. accepted
DOI: 
7 Electrochemical Synthesis of Heterodehydro[7]helicenes
Khalid Md. Imrul, Salem M. S. H., Sako Makoto, Kondo Masaru, Sasai Hiroaki*, Takizawa Shinobu*
Commun. Chem. accepted
DOI: 
8 Total Synthesis of Ansellone G and Phorbadione
Yanagihara Mizushi, Nakahara Kanae, Kishimoto Naoki, Abe Towa, Miura Satoshi, Misumi Shogo, Sako Makoto, Arisawa Mitsuhiro* Murai Kenichi*
J. Org. Chem. accepted
DOI: 
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Ⅱ. Review
1 環境調和型非イオン性両親媒性化合物を用いる水中金属触媒反応
和田 祐希
ファルマシア, Vol. 58, No.3 (2022), 261.
DOI: 10.14894/10.14894/faruawpsj.58.3_261
   
   
Ⅲ. Winning Prize
1 大阪大学沢井記念薬友会賞スタートアップ賞
渡邊君(B4)が大阪大学沢井記念薬友会賞スタートアップ賞を受賞しました。
2

第72回日本薬学会関西支部総会・大会 優秀ポスター発表賞
髙島さん(B4)が第72回日本薬学会関西支部総会・大会優秀ポスター発表賞を受賞しました。

    
   
Ⅳ. その他
1 [研究室紹介]有澤研究室(阪大院薬)
Organometallic News, No. 3 (2022), 85-86.
https://kinka.or.jp/om/omnews_archive/2022_03.html